lol lol lol lol wrote:
GoldenMiles wrote:Interesting. Why Tramadol and not more traditional opiates (hydrocodone, oxycodone, morphine, etc.)? I'm guessing they abuse it to stop the pain of hard athletic efforts?
If other opioids are banned and tramadol is not, that would be one reason--I'd google to see if this is the case.
Tramadol is also not merely an opioid; it is an extremely weird drug which functions as
1) A very weak opioid
2) A prodrug which is converted in the liver into a much stronger opioid
3) An SNRI, a la Venlafaxine (Effexor)
4) A serotonin-releasing agent, a la MDMA (Ecstasy)
There are other effects as well...
The effect on norepinephrine makes tramadol much more stimulating than pure opioids, this is advantageous to endurance athletes.
One thing I will say to those looking to abuse Tramadol (I've done it a few times when I had a low opiate tolerance, and it does give a nice, relaxing high), I've heard many say that it has worse withdrawals than comparable opiates in strength (hydrocodone, codeine, etc.), because, as mentioned by lol lol lol, it is both an opioid (not sure if it's technically an opiate) and an anti-depressant (an SNRI, as listed above). You will get both opiate withdrawals and anti-depressant withdrawals upon stopping taking it.
Not sure about this part, but if it is heavily drawing upon your serotonin, you might feel an awful crash similar to if you do too much Ecstasy, which leaves your brain and emotions feeling sapped (never did too much MDMA myself, since it never made me feel that good, surprisingly).
It makes sense if athletes would take it if it isn't banned or doesn't show up on drug tests. For instance, Suboxone doesn't show up on most drug tests I've taken as an opiate, since it's structurally close but still dissimilar to something like heroin/morphine, oxy/hydrocodone, codeine, or hydromorphone (Dilaudid).